Giosuè Costa

InstitutionUniversità 'Magna Græcia'
AddressCatanzaro
Italy
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    Publication Timeline
    COVID-19 publications
    Bar chart showing 2 Covid-19 publications, with a maximum of 1 publications in August 2020 and January 2021
    All Publications
    Bar chart showing 49 publications over 12 distinct years, with a maximum of 8 publications in 2016
    These graphs show COVID-19 publications by month since August 2019 and all publications written by authors of COVID-19 publications over the past 30 years.

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    Publication Field Summary
    This graph shows the number and percent of publications by field. Fields are based on how the National Library of Medicine (NLM) classifies the publications' journals and might not represent the specific topics of the publications. Note that an individual publication can be assigned to more than one field. As a result, the publication counts in this graph might add up to more than the number of publications the person has written. To see the data as text, click here.
    Publication List
    Publications listed below are automatically derived from MEDLINE/PubMed and other sources, which might result in incorrect or missing publications.
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    PMC Citations indicate the number of times the publication was cited by articles in PubMed Central, and the Altmetric score represents citations in news articles and social media. (Note that publications are often cited in additional ways that are not shown here.) Fields are based on how the National Library of Medicine (NLM) classifies the publication's journal and might not represent the specific topic of the publication. Translation tags are based on the publication type and the MeSH terms NLM assigns to the publication. Some publications (especially newer ones and publications not in PubMed) might not yet be assigned Field or Translation tags.) Click a Field or Translation tag to filter the publications.
    1. Salpini R, Alkhatib M, Costa G, Piermatteo L, Ambrosio FA, Di Maio VC, Scutari R, Duca L, Berno G, Fabeni L, Alcaro S, Ceccherini-Silberstein F, Artese A, Svicher V. Key genetic elements, single and in clusters, underlying geographically dependent SARS-CoV-2 genetic adaptation and their impact on binding affinity for drugs and immune control. J Antimicrob Chemother. 2021 01 19; 76(2):396-412. PMID: 33254234.
      Citations: 4     Fields:    Translation:HumansCells
    2. Artese A, Svicher V, Costa G, Salpini R, Di Maio VC, Alkhatib M, Ambrosio FA, Santoro MM, Assaraf YG, Alcaro S, Ceccherini-Silberstein F. Current status of antivirals and druggable targets of SARS CoV-2 and other human pathogenic coronaviruses. Drug Resist Updat. 2020 12; 53:100721. PMID: 33132205.
      Citations: 20     Fields:    Translation:HumansAnimalsCells
    3. Maruca A, Catalano R, Bagetta D, Mesiti F, Ambrosio FA, Romeo I, Moraca F, Rocca R, Ortuso F, Artese A, Costa G, Alcaro S, Lupia A. The Mediterranean Diet as source of bioactive compounds with multi-targeting anti-cancer profile. Eur J Med Chem. 2019 Nov 01; 181:111579. PMID: 31398616.
      Citations: 13     Fields:    Translation:HumansAnimals
    4. Costa G, Carta F, Ambrosio FA, Artese A, Ortuso F, Moraca F, Rocca R, Romeo I, Lupia A, Maruca A, Bagetta D, Catalano R, Vullo D, Alcaro S, Supuran CT. A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors. Eur J Med Chem. 2019 Nov 01; 181:111565. PMID: 31387062.
      Citations: 8     Fields:    Translation:Humans
    5. Costa G, Rocca R, Corona A, Grandi N, Moraca F, Romeo I, Talarico C, Gagliardi MG, Ambrosio FA, Ortuso F, Alcaro S, Distinto S, Maccioni E, Tramontano E, Artese A. Novel natural non-nucleoside inhibitors of HIV-1 reverse transcriptase identified by shape- and structure-based virtual screening techniques. Eur J Med Chem. 2019 Jan 01; 161:1-10. PMID: 30342421.
      Citations: 14     Fields:    Translation:HumansCells
    6. Vasile F, Della Volpe S, Ambrosio FA, Costa G, Unver MY, Zucal C, Rossi D, Martino E, Provenzani A, Hirsch AKH, Alcaro S, Potenza D, Collina S. Exploration of ligand binding modes towards the identification of compounds targeting HuR: a combined STD-NMR and Molecular Modelling approach. Sci Rep. 2018 09 13; 8(1):13780. PMID: 30214075.
      Citations: 4     Fields:    Translation:HumansCells
    7. Rocca R, Moraca F, Costa G, Talarico C, Ortuso F, Da Ros S, Nicoletto G, Sissi C, Alcaro S, Artese A. In Silico Identification of Piperidinyl-amine Derivatives as Novel Dual Binders of Oncogene c-myc/c-Kit G-quadruplexes. ACS Med Chem Lett. 2018 Aug 09; 9(8):848-853. PMID: 30128079.
      Citations: 6     
    8. Malet I, Ambrosio FA, Subra F, Herrmann B, Leh H, Bouger MC, Artese A, Katlama C, Talarico C, Romeo I, Alcaro S, Costa G, Deprez E, Calvez V, Marcelin AG, Delelis O. Pathway involving the N155H mutation in HIV-1 integrase leads to dolutegravir resistance. J Antimicrob Chemother. 2018 05 01; 73(5):1158-1166. PMID: 29373677.
      Citations: 5     Fields:    Translation:HumansCells
    9. Gaudio E, Paduano F, Pinton S, D'Agostino S, Rocca R, Costa G, Ngankeu A, Aqeilan RI, Croce CM, Bertoni F, Alcaro S, Trapasso F. TCL1A interacts with TP63 and enhances the survival of Raji Burkitt lymphoma cell line. Br J Haematol. 2018 11; 183(3):509-512. PMID: 29048125.
      Citations: 3     Fields:    Translation:HumansCells
    10. Rocca R, Talarico C, Moraca F, Costa G, Romeo I, Ortuso F, Alcaro S, Artese A. Molecular recognition of a carboxy pyridostatin toward G-quadruplex structures: Why does it prefer RNA? Chem Biol Drug Des. 2017 Nov; 90(5):919-925. PMID: 28459507.
      Citations: 7     Fields:    Translation:Cells
    11. Milelli A, Marchetti C, Greco ML, Moraca F, Costa G, Turrini E, Catanzaro E, Betari N, Calcabrini C, Sissi C, Alcaro S, Fimognari C, Tumiatti V, Minarini A. Naphthalene diimide-polyamine hybrids as antiproliferative agents: Focus on the architecture of the polyamine chains. Eur J Med Chem. 2017 Mar 10; 128:107-122. PMID: 28157593.
      Citations: 4     Fields:    Translation:HumansCells
    12. Rocca R, Moraca F, Costa G, Nadai M, Scalabrin M, Talarico C, Distinto S, Maccioni E, Ortuso F, Artese A, Alcaro S, Richter SN. Identification of G-quadruplex DNA/RNA binders: Structure-based virtual screening and biophysical characterization. Biochim Biophys Acta Gen Subj. 2017 May; 1861(5 Pt B):1329-1340. PMID: 28025082.
      Citations: 13     Fields:    Translation:Cells
    13. Carradori S, Gidaro MC, Petzer A, Costa G, Guglielmi P, Chimenti P, Alcaro S, Petzer JP. Inhibition of Human Monoamine Oxidase: Biological and Molecular Modeling Studies on Selected Natural Flavonoids. J Agric Food Chem. 2016 Nov 30; 64(47):9004-9011. PMID: 27933876.
      Citations: 11     Fields:    Translation:Humans
    14. Alteri C, Surdo M, Di Maio VC, Di Santo F, Costa G, Parrotta L, Romeo I, Gori C, Santoro MM, Fedele V, Carta S, Continenza F, Pinnetti C, Bellagamba R, Liuzzi G, Orchi N, Latini A, Bertoli A, Girardi E, Alcaro S, Giuliani M, Petrosillo N, Andreoni M, Antinori A, Monforte AD, Ceccherini-Silberstein F, Artese A, Perno CF, Svicher V. The HIV-1 reverse transcriptase polymorphism A98S improves the response to tenofovir disoproxil fumarate+emtricitabine-containing HAART both in vivo and in vitro. J Glob Antimicrob Resist. 2016 12; 7:1-7. PMID: 27530997.
      Citations: 1     Fields:    Translation:HumansCells
    15. Costa G, Rocca R, Moraca F, Talarico C, Romeo I, Ortuso F, Alcaro S, Artese A. A Comparative Docking Strategy to Identify Polyphenolic Derivatives as Promising Antineoplastic Binders of G-quadruplex DNA c-myc and bcl-2 Sequences. Mol Inform. 2016 09; 35(8-9):391-402. PMID: 27546043.
      Citations: 5     Fields:    Translation:HumansCells
    16. Costa G, Gidaro MC, Vullo D, Supuran CT, Alcaro S. Active Components of Essential Oils as Anti-Obesity Potential Drugs Investigated by in Silico Techniques. J Agric Food Chem. 2016 Jul 06; 64(26):5295-300. PMID: 27268752.
      Citations: 5     Fields:    Translation:HumansCells
    17. Varela CL, Amaral C, Correia-da-Silva G, Costa SC, Carvalho RA, Costa G, Alcaro S, Teixeira NA, Tavares-da-Silva EJ, Roleira FM. Exploring new chemical functionalities to improve aromatase inhibition of steroids. Bioorg Med Chem. 2016 06 15; 24(12):2823-31. PMID: 27160054.
      Citations:    Fields:    Translation:HumansCells
    18. Rocca R, Costa G, Artese A, Parrotta L, Ortuso F, Maccioni E, Pinato O, Greco ML, Sissi C, Alcaro S, Distinto S, Moraca F. Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement. ChemMedChem. 2016 08 19; 11(16):1721-33. PMID: 27008476.
      Citations: 8     Fields:    Translation:HumansCells
    19. Gidaro MC, Astorino C, Petzer A, Carradori S, Alcaro F, Costa G, Artese A, Rafele G, Russo FM, Petzer JP, Alcaro S. Kaempferol as Selective Human MAO-A Inhibitor: Analytical Detection in Calabrian Red Wines, Biological and Molecular Modeling Studies. J Agric Food Chem. 2016 Feb 17; 64(6):1394-400. PMID: 26821152.
      Citations: 11     Fields:    Translation:Humans
    20. D'Ascenzio M, Chimenti P, Gidaro MC, De Monte C, De Vita D, Granese A, Scipione L, Di Santo R, Costa G, Alcaro S, Yáñez M, Carradori S. (Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies. J Enzyme Inhib Med Chem. 2015 Dec; 30(6):908-19. PMID: 25807300.
      Citations: 2     Fields:    Translation:HumansCells
    21. De Monte C, Bizzarri B, Gidaro MC, Carradori S, Mollica A, Luisi G, Granese A, Alcaro S, Costa G, Basilico N, Parapini S, Scaltrito MM, Masia C, Sisto F. Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents. J Enzyme Inhib Med Chem. 2015 Dec; 30(6):1027-33. PMID: 25766747.
      Citations: 9     Fields:    Translation:AnimalsCells
    22. Alteri C, Surdo M, Bellocchi MC, Saccomandi P, Continenza F, Armenia D, Parrotta L, Carioti L, Costa G, Fourati S, Di Santo F, Scutari R, Barbaliscia S, Fedele V, Carta S, Balestra E, Alcaro S, Marcelin AG, Calvez V, Ceccherini-Silberstein F, Artese A, Perno CF, Svicher V. Incomplete APOBEC3G/F Neutralization by HIV-1 Vif Mutants Facilitates the Genetic Evolution from CCR5 to CXCR4 Usage. Antimicrob Agents Chemother. 2015 Aug; 59(8):4870-81. PMID: 26055363.
      Citations: 7     Fields:    Translation:HumansCells
    23. D'Antona L, Amato R, Talarico C, Ortuso F, Menniti M, Dattilo V, Iuliano R, Gigliotti F, Artese A, Costa G, Schenone S, Musumeci F, Abbruzzese C, Botta L, Trapasso F, Alcaro S, Paggi MG, Perrotti N. SI113, a specific inhibitor of the Sgk1 kinase activity that counteracts cancer cell proliferation. Cell Physiol Biochem. 2015; 35(5):2006-18. PMID: 25871776.
      Citations: 21     Fields:    Translation:HumansCells
    24. Gidaro MC, Alcaro F, Carradori S, Costa G, Vullo D, Supuran CT, Alcaro S. Erratum for: Eriocitrin and Apigenin as New Carbonic Anhydrase VA Inhibitors from a Virtual Screening of Calabrian Natural Products. Planta Med. 2015 04; 81(6):E1. PMID: 25625199.
      Citations:    Fields:    
    25. Gidaro MC, Alcaro F, Carradori S, Costa G, Vullo D, Supuran CT, Alcaro S. Eriocitrin and Apigenin as New Carbonic Anhydrase VA Inhibitors from a Virtual Screening of Calabrian Natural Products. Planta Med. 2015 Apr; 81(6):533-40. PMID: 25590364.
      Citations: 3     Fields:    Translation:Animals
    26. Rocca R, Moraca F, Costa G, Alcaro S, Distinto S, Maccioni E, Ortuso F, Artese A, Parrotta L. Structure-based virtual screening of novel natural alkaloid derivatives as potential binders of h-telo and c-myc DNA G-quadruplex conformations. Molecules. 2014 Dec 24; 20(1):206-23. PMID: 25547724.
      Citations: 9     Fields:    Translation:HumansCells
    27. Parrotta L, Ortuso F, Moraca F, Rocca R, Costa G, Alcaro S, Artese A. Targeting unimolecular G-quadruplex nucleic acids: a new paradigm for the drug discovery? Expert Opin Drug Discov. 2014 Oct; 9(10):1167-87. PMID: 25109710.
      Citations: 8     Fields:    Translation:HumansCells
    28. Ortuso F, Amato R, Artese A, D'antona L, Costa G, Talarico C, Gigliotti F, Bianco C, Trapasso F, Schenone S, Musumeci F, Botta L, Perrotti N, Alcaro S. In silico identification and biological evaluation of novel selective serum/glucocorticoid-inducible kinase 1 inhibitors based on the pyrazolo-pyrimidine scaffold. J Chem Inf Model. 2014 Jul 28; 54(7):1828-32. PMID: 24896223.
      Citations: 20     Fields:    Translation:HumansCells
    29. De Monte C, Carradori S, Chimenti P, Secci D, Mannina L, Alcaro F, Petzer A, N'Da CI, Gidaro MC, Costa G, Alcaro S, Petzer JP. New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies. Eur J Med Chem. 2014 Jul 23; 82:164-71. PMID: 24904963.
      Citations: 9     Fields:    Translation:HumansAnimalsCells
    30. Percivalle C, Sissi C, Greco ML, Musetti C, Mariani A, Artese A, Costa G, Perrore ML, Alcaro S, Freccero M. Aryl ethynyl anthraquinones: a useful platform for targeting telomeric G-quadruplex structures. Org Biomol Chem. 2014 Jun 14; 12(22):3744-54. PMID: 24789544.
      Citations: 1     Fields:    Translation:Cells
    31. Malet I, Gimferrer Arriaga L, Artese A, Costa G, Parrotta L, Alcaro S, Delelis O, Tmeizeh A, Katlama C, Valantin MA, Ceccherini-Silberstein F, Calvez V, Marcelin AG. New raltegravir resistance pathways induce broad cross-resistance to all currently used integrase inhibitors. J Antimicrob Chemother. 2014 Aug; 69(8):2118-22. PMID: 24710029.
      Citations: 25     Fields:    Translation:HumansCells
    32. Sattin G, Artese A, Nadai M, Costa G, Parrotta L, Alcaro S, Palumbo M, Richter SN. Conformation and stability of intramolecular telomeric G-quadruplexes: sequence effects in the loops. PLoS One. 2013; 8(12):e84113. PMID: 24367632.
      Citations: 10     Fields:    Translation:HumansCells
    33. Artese A, Costa G, Ortuso F, Parrotta L, Alcaro S. Identification of new natural DNA G-quadruplex binders selected by a structure-based virtual screening approach. Molecules. 2013 Sep 30; 18(10):12051-70. PMID: 24084014.
      Citations: 5     Fields:    Translation:HumansCells
    34. Artese A, Costa G, Distinto S, Moraca F, Ortuso F, Parrotta L, Alcaro S. Toward the design of new DNA G-quadruplex ligands through rational analysis of polymorphism and binding data. Eur J Med Chem. 2013 Oct; 68:139-49. PMID: 23974014.
      Citations: 3     Fields:    Translation:HumansCells
    35. Fourati S, Visseaux B, Armenia D, Morand-Joubert L, Artese A, Charpentier C, Van Den Eede P, Costa G, Alcaro S, Wirden M, Perno CF, Ceccherini Silberstein F, Descamps D, Calvez V, Marcelin AG. Identification of a rare mutation at reverse transcriptase Lys65 (K65E) in HIV-1-infected patients failing on nucleos(t)ide reverse transcriptase inhibitors. J Antimicrob Chemother. 2013 Oct; 68(10):2199-204. PMID: 23749955.
      Citations: 5     Fields:    Translation:HumansCells
    36. Alteri C, Artese A, Beheydt G, Santoro MM, Costa G, Parrotta L, Bertoli A, Gori C, Orchi N, Girardi E, Antinori A, Alcaro S, d'Arminio Monforte A, Theys K, Vandamme AM, Ceccherini-Silberstein F, Svicher V, Perno CF. Structural modifications induced by specific HIV-1 protease-compensatory mutations have an impact on the virological response to a first-line lopinavir/ritonavir-containing regimen. J Antimicrob Chemother. 2013 Oct; 68(10):2205-9. PMID: 23687186.
      Citations: 3     Fields:    Translation:HumansCells
    37. Alcaro S, Musetti C, Distinto S, Casatti M, Zagotto G, Artese A, Parrotta L, Moraca F, Costa G, Ortuso F, Maccioni E, Sissi C. Identification and characterization of new DNA G-quadruplex binders selected by a combination of ligand and structure-based virtual screening approaches. J Med Chem. 2013 Feb 14; 56(3):843-55. PMID: 23294188.
      Citations: 21     Fields:    Translation:Cells
    38. Chen M, Svicher V, Artese A, Costa G, Alteri C, Ortuso F, Parrotta L, Liu Y, Liu C, Perno CF, Alcaro S, Zhang J. Detecting and understanding genetic and structural features in HIV-1 B subtype V3 underlying HIV-1 co-receptor usage. Bioinformatics. 2013 Feb 15; 29(4):451-60. PMID: 23297034.
      Citations: 7     Fields:    Translation:HumansCells
    39. Cross S, Ortuso F, Baroni M, Costa G, Distinto S, Moraca F, Alcaro S, Cruciani G. GRID-based three-dimensional pharmacophores II: PharmBench, a benchmark data set for evaluating pharmacophore elucidation methods. J Chem Inf Model. 2012 Oct 22; 52(10):2599-608. PMID: 22970854.
      Citations: 5     Fields:    Translation:HumansCells
    40. Cento V, Mirabelli C, Salpini R, Dimonte S, Artese A, Costa G, Mercurio F, Svicher V, Parrotta L, Bertoli A, Ciotti M, Di Paolo D, Sarrecchia C, Andreoni M, Alcaro S, Angelico M, Perno CF, Ceccherini-Silberstein F. HCV genotypes are differently prone to the development of resistance to linear and macrocyclic protease inhibitors. PLoS One. 2012; 7(7):e39652. PMID: 22792183.
      Citations: 31     Fields:    Translation:HumansCells
    41. Varela C, Tavares da Silva EJ, Amaral C, Correia da Silva G, Baptista T, Alcaro S, Costa G, Carvalho RA, Teixeira NA, Roleira FM. New structure-activity relationships of A- and D-ring modified steroidal aromatase inhibitors: design, synthesis, and biochemical evaluation. J Med Chem. 2012 Apr 26; 55(8):3992-4002. PMID: 22475216.
      Citations: 9     Fields:    Translation:HumansCells
    42. Alcaro S, Alteri C, Artese A, Ceccherini-Silberstein F, Costa G, Ortuso F, Bertoli A, Forbici F, Santoro MM, Parrotta L, Flandre P, Masquelier B, Descamps D, Calvez V, Marcelin AG, Perno CF, Sing T, Svicher V. Docking analysis and resistance evaluation of clinically relevant mutations associated with the HIV-1 non-nucleoside reverse transcriptase inhibitors nevirapine, efavirenz and etravirine. ChemMedChem. 2011 Dec 09; 6(12):2203-13. PMID: 21953939.
      Citations: 8     Fields:    Translation:HumansCells
    43. Maccioni E, Alcaro S, Cirilli R, Vigo S, Cardia MC, Sanna ML, Meleddu R, Yanez M, Costa G, Casu L, Matyus P, Distinto S. 3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B. J Med Chem. 2011 Sep 22; 54(18):6394-8. PMID: 21777011.
      Citations: 8     Fields:    Translation:HumansAnimalsCells
    44. Alcaro S, Artese A, Costa G, Distinto S, Ortuso F, Parrotta L. Conformational studies and solvent-accessible surface area analysis of known selective DNA G-Quadruplex binders. Biochimie. 2011 Aug; 93(8):1267-74. PMID: 21699954.
      Citations: 3     Fields:    Translation:HumansCells
    45. Alcaro S, Alteri C, Artese A, Ceccherini-Silberstein F, Costa G, Ortuso F, Parrotta L, Perno CF, Svicher V. Molecular and structural aspects of clinically relevant mutations related to the approved non-nucleoside inhibitors of HIV-1 reverse transcriptase. Drug Resist Updat. 2011 Jun; 14(3):141-9. PMID: 21295512.
      Citations: 3     Fields:    Translation:HumansCells
    46. Svicher V, Alteri C, Artese A, Zhang JM, Costa G, Mercurio F, D'Arrigo R, Alcaro S, Palù G, Clementi M, Zazzi M, Andreoni M, Antinori A, Lazzarin A, Ceccherini-Silberstein F, Perno CF. Identification and structural characterization of novel genetic elements in the HIV-1 V3 loop regulating coreceptor usage. Antivir Ther. 2011; 16(7):1035-45. PMID: 22024519.
      Citations: 9     Fields:    Translation:HumansCells
    47. Svicher V, Alteri C, Artese A, Forbici F, Santoro MM, Schols D, Van Laethem K, Alcaro S, Costa G, Tommasi C, Zaccarelli M, Narciso P, Antinori A, Ceccherini-Silberstein F, Balzarini J, Perno CF. Different evolution of genotypic resistance profiles to emtricitabine versus lamivudine in tenofovir-containing regimens. J Acquir Immune Defic Syndr. 2010 Nov; 55(3):336-44. PMID: 20739898.
      Citations: 8     Translation:HumansCells
    48. Ceccherini-Silberstein F, Malet I, Fabeni L, Dimonte S, Svicher V, D'Arrigo R, Artese A, Costa G, Bono S, Alcaro S, Monforte Ad, Katlama C, Calvez V, Antinori A, Marcelin AG, Perno CF. Specific HIV-1 integrase polymorphisms change their prevalence in untreated versus antiretroviral-treated HIV-1-infected patients, all naive to integrase inhibitors. J Antimicrob Chemother. 2010 Nov; 65(11):2305-18. PMID: 20817922.
      Citations: 24     Fields:    Translation:HumansCells
    49. Alcaro S, Arcone R, Costa G, De Vita D, Iannone M, Ortuso F, Procopio A, Pasceri R, Rotiroti D, Scipione L. Simple choline esters as potential anti-Alzheimer agents. Curr Pharm Des. 2010; 16(6):692-7. PMID: 20388079.
      Citations: 2     Fields:    Translation:AnimalsCells