Wolfgang Holzer

InstitutionUniversity of Vienna
AddressAustria
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    Publication Timeline
    COVID-19 publications
    Bar chart showing 1 Covid-19 publications, with a maximum of 1 publications in January 2021
    All Publications
    Bar chart showing 62 publications over 18 distinct years, with a maximum of 10 publications in 2016
    These graphs show COVID-19 publications by month since August 2019 and all publications written by authors of COVID-19 publications over the past 30 years.

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    Publication Field Summary
    This graph shows the number and percent of publications by field. Fields are based on how the National Library of Medicine (NLM) classifies the publications' journals and might not represent the specific topics of the publications. Note that an individual publication can be assigned to more than one field. As a result, the publication counts in this graph might add up to more than the number of publications the person has written. To see the data as text, click here.
    Publication List
    Publications listed below are automatically derived from MEDLINE/PubMed and other sources, which might result in incorrect or missing publications.
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    PMC Citations indicate the number of times the publication was cited by articles in PubMed Central, and the Altmetric score represents citations in news articles and social media. (Note that publications are often cited in additional ways that are not shown here.) Fields are based on how the National Library of Medicine (NLM) classifies the publication's journal and might not represent the specific topic of the publication. Translation tags are based on the publication type and the MeSH terms NLM assigns to the publication. Some publications (especially newer ones and publications not in PubMed) might not yet be assigned Field or Translation tags.) Click a Field or Translation tag to filter the publications.
    1. Citarella A, Gentile D, Rescifina A, Piperno A, Mognetti B, Gribaudo G, Sciortino MT, Holzer W, Pace V, Micale N. Pseudo-Dipeptide Bearing a,a-Difluoromethyl Ketone Moiety as Electrophilic Warhead with Activity against Coronaviruses. Int J Mol Sci. 2021 Jan 30; 22(3). PMID: 33573283.
      Citations: 3     Fields:    Translation:HumansCells
    2. Miele M, D'Orsi R, Sridharan V, Holzer W, Pace V. Highly chemoselective difluoromethylative homologation of iso(thio)cyanates: expeditious access to unprecedented a,a-difluoro(thio)amides. Chem Commun (Camb). 2019 Oct 24; 55(86):12960-12963. PMID: 31602439.
      Citations: 3     Fields:    
    3. Pace V, Holzer W, Ielo L, Shi S, Meng G, Hanna M, Szostak R, Szostak M. 17O NMR and 15N NMR chemical shifts of sterically-hindered amides: ground-state destabilization in amide electrophilicity. Chem Commun (Camb). 2019 Apr 09; 55(30):4423-4426. PMID: 30916689.
      Citations: 1     Fields:    
    4. Milišiunaite V, Paulaviciute R, Arbaciauskiene E, Martynaitis V, Holzer W, Šackus A. Synthesis of 2H-furo[2,3-c]pyrazole ring systems through silver(I) ion-mediated ring-closure reaction. Beilstein J Org Chem. 2019; 15:679-684. PMID: 30931008.
      Citations: 2     
    5. Monticelli S, Holzer W, Langer T, Roller A, Olofsson B, Pace V. Sustainable Asymmetric Organolithium Chemistry: Enantio- and Chemoselective Acylations through Recycling of Solvent, Sparteine, and Weinreb "Amine". ChemSusChem. 2019 Mar 21; 12(6):1147-1154. PMID: 30614208.
      Citations: 2     Fields:    
    6. de la Vega-Hernández K, Senatore R, Miele M, Urban E, Holzer W, Pace V. Chemoselective reduction of isothiocyanates to thioformamides mediated by the Schwartz reagent. Org Biomol Chem. 2019 02 13; 17(7):1970-1978. PMID: 30362485.
      Citations: 2     Fields:    
    7. Monticelli S, Colella M, Pillari V, Tota A, Langer T, Holzer W, Degennaro L, Luisi R, Pace V. Modular and Chemoselective Strategy for the Direct Access to a-Fluoroepoxides and Aziridines via the Addition of Fluoroiodomethyllithium to Carbonyl-Like Compounds. Org Lett. 2019 01 18; 21(2):584-588. PMID: 30600682.
      Citations: 7     Fields:    
    8. Stadler M, Monticelli S, Seidel T, Luger D, Salzer I, Boehm S, Holzer W, Schwarzer C, Urban E, Khom S, Langer T, Pace V, Hering S. Design, Synthesis, and Pharmacological Evaluation of Novel ß2/3 Subunit-Selective ?-Aminobutyric Acid Type A (GABAA) Receptor Modulators. J Med Chem. 2019 01 10; 62(1):317-341. PMID: 30289721.
      Citations: 2     Fields:    Translation:AnimalsCells
    9. Touqeer S, Castoldi L, Langer T, Holzer W, Pace V. Homologation of halostannanes with carbenoids: a convenient and straightforward one-step access to a-functionalized organotin reagents. Chem Commun (Camb). 2018 Sep 06; 54(72):10112-10115. PMID: 30124702.
      Citations: 1     Fields:    
    10. Eller GA, Vilkauskaite G, Šackus A, Martynaitis V, Mamuye AD, Pace V, Holzer W. An unusual thionyl chloride-promoted C-C bond formation to obtain 4,4'-bipyrazolones. Beilstein J Org Chem. 2018; 14:1287-1292. PMID: 29977396.
      Citations: 1     
    11. Senatore R, Castoldi L, Ielo L, Holzer W, Pace V. Expeditious and Chemoselective Synthesis of a-Aryl and a-Alkyl Selenomethylketones via Homologation Chemistry. Org Lett. 2018 05 04; 20(9):2685-2688. PMID: 29664309.
      Citations: 4     Fields:    
    12. Castoldi L, Ielo L, Holzer W, Giester G, Roller A, Pace V. a-Arylamino Diazoketones: Diazomethane-Loading Controlled Synthesis, Spectroscopic Investigations, and Structural X-ray Analysis. J Org Chem. 2018 04 20; 83(8):4336-4347. PMID: 29546992.
      Citations: 1     Fields:    
    13. Milišiunaite V, Arbaciauskiene E, Reznícková E, Jorda R, Malínková V, Žukauskaite A, Holzer W, Šackus A, Kryštof V. Synthesis and anti-mitotic activity of 2,4- or 2,6-disubstituted- and 2,4,6-trisubstituted-2H-pyrazolo[4,3-c]pyridines. Eur J Med Chem. 2018 Apr 25; 150:908-919. PMID: 29602037.
      Citations: 3     Fields:    Translation:HumansCells
    14. Arbaciauskiene E, Krikštolaityte S, Mitruleviciene A, Bieliauskas A, Martynaitis V, Bechmann M, Roller A, Šackus A, Holzer W. On the Tautomerism of N-Substituted Pyrazolones: 1,2-Dihydro-3H-pyrazol-3-ones versus 1H-Pyrazol-3-ols. Molecules. 2018 Jan 09; 23(1). PMID: 29315238.
      Citations: 2     Fields:    Translation:Cells
    15. Parisi G, Colella M, Monticelli S, Romanazzi G, Holzer W, Langer T, Degennaro L, Pace V, Luisi R. Exploiting a "Beast" in Carbenoid Chemistry: Development of a Straightforward Direct Nucleophilic Fluoromethylation Strategy. J Am Chem Soc. 2017 10 04; 139(39):13648-13651. PMID: 28892363.
      Citations: 13     Fields:    
    16. Pace V, Castoldi L, Mazzeo E, Rui M, Langer T, Holzer W. Efficient Access to All-Carbon Quaternary and Tertiary a-Functionalized Homoallyl-type Aldehydes from Ketones. Angew Chem Int Ed Engl. 2017 10 02; 56(41):12677-12682. PMID: 28722252.
      Citations: 7     Fields:    
    17. Castoldi L, Holzer W, Langer T, Pace V. Evidence and isolation of tetrahedral intermediates formed upon the addition of lithium carbenoids to Weinreb amides and N-acylpyrroles. Chem Commun (Camb). 2017 Aug 22; 53(68):9498-9501. PMID: 28799583.
      Citations: 4     Fields:    
    18. Parisi G, Degennaro L, Carlucci C, de Candia M, Mastrorilli P, Roller A, Holzer W, Altomare CD, Pace V, Luisi R. A greener and efficient access to substituted four- and six-membered sulfur-bearing heterocycles. Org Biomol Chem. 2017 Jun 14; 15(23):5000-5015. PMID: 28567461.
      Citations: 2     Fields:    
    19. Jansa J, Schmidt R, Mamuye AD, Castoldi L, Roller A, Pace V, Holzer W. Synthesis of tetrasubstituted pyrazoles containing pyridinyl substituents. Beilstein J Org Chem. 2017; 13:895-902. PMID: 28546847.
      Citations: 1     
    20. Pace V, Holzer W, Meng G, Shi S, Lalancette R, Szostak R, Szostak M. Corrigendum: Structures of Highly Twisted Amides Relevant to Amide N-C Cross-Coupling: Evidence for Ground-State Amide Destabilization. Chemistry. 2017 03 08; 23(14):3496. PMID: 28276655.
      Citations:    Fields:    
    21. Schuster R, Zeindl L, Holzer W, Khumpirapang N, Okonogi S, Viernstein H, Mueller M. Eulophia macrobulbon - an orchid with significant anti-inflammatory and antioxidant effect and anticancerogenic potential exerted by its root extract. Phytomedicine. 2017 Jan 15; 24:157-165. PMID: 28160857.
      Citations: 5     Fields:    Translation:HumansAnimalsCells
    22. Praznik W, Cavarkapa A, Unger FM, Loeppert R, Holzer W, Viernstein H, Mueller M. Molecular dimensions and structural features of neutral polysaccharides from the seed mucilage of Hyptis suaveolens L. Food Chem. 2017 Apr 15; 221:1997-2004. PMID: 27979191.
      Citations: 1     Fields:    Translation:AnimalsCells
    23. Okonogi S, Kheawfu K, Holzer W, Unger FM, Viernstein H, Mueller M. Anti-inflammatory Effects of Compounds from Polygonum odoratum. Nat Prod Commun. 2016 Nov; 11(11):1651-1654. PMID: 30475499.
      Citations: 3     Fields:    Translation:AnimalsCells
    24. Monticelli S, Parisi G, Rui M, de la Vega-Hernández K, Murgia I, Senatore R, Holzer W, Urban E, Langer T, Pace V. The Use of the Comins-Meyers Amide in Synthetic Chemistry: an Overview. Nat Prod Commun. 2016 Nov; 11(11):1729-1732. PMID: 30475518.
      Citations:    Fields:    Translation:Cells
    25. Schuster R, Holzer W, Doerfler H, Weckwerth W, Viernstein H, Okonogi S, Mueller M. Cajanus cajan- a source of PPAR? activators leading to anti-inflammatory and cytotoxic effects. Food Funct. 2016 Sep 14; 7(9):3798-806. PMID: 27603115.
      Citations: 2     Fields:    Translation:HumansAnimalsCells
    26. Pace V, Holzer W, Meng G, Shi S, Lalancette R, Szostak R, Szostak M. Structures of Highly Twisted Amides Relevant to Amide N-C Cross-Coupling: Evidence for Ground-State Amide Destabilization. Chemistry. 2016 Oct 04; 22(41):14494-8. PMID: 27558185.
      Citations: 5     Fields:    
    27. Pace V, Holzer W, De Kimpe N. Lithium Halomethylcarbenoids: Preparation and Use in the Homologation of Carbon Electrophiles. Chem Rec. 2016 08; 16(4):2061-76. PMID: 27381551.
      Citations: 6     Fields:    
    28. Pace V, Murgia I, Westermayer S, Langer T, Holzer W. Highly efficient synthesis of functionalized a-oxyketones via Weinreb amides homologation with a-oxygenated organolithiums. Chem Commun (Camb). 2016 Jun 18; 52(48):7584-7. PMID: 27220327.
      Citations: 5     Fields:    
    29. Mueller M, Weinmann D, Toegel S, Holzer W, Unger FM, Viernstein H. Compounds from Caesalpinia sappan with anti-inflammatory properties in macrophages and chondrocytes. Food Funct. 2016 Mar; 7(3):1671-9. PMID: 26951869.
      Citations: 7     Fields:    Translation:HumansAnimalsCells
    30. Pace V, Pelosi A, Antermite D, Rosati O, Curini M, Holzer W. Bromomethyllithium-mediated chemoselective homologation of disulfides to dithioacetals. Chem Commun (Camb). 2016 Feb 11; 52(12):2639-42. PMID: 26750866.
      Citations: 4     Fields:    
    31. Pace V, Castoldi L, Monticelli S, Safranek S, Roller A, Langer T, Holzer W. A Robust, Eco-Friendly Access to Secondary Thioamides through the Addition of Organolithium Reagents to Isothiocyanates in Cyclopentyl Methyl Ether (CPME). Chemistry. 2015 Dec 21; 21(52):18966-70. PMID: 26507565.
      Citations: 3     Fields:    
    32. Mamuye AD, Castoldi L, Azzena U, Holzer W, Pace V. Chemoselective efficient synthesis of functionalized ß-oxonitriles through cyanomethylation of Weinreb amides. Org Biomol Chem. 2015 Feb 21; 13(7):1969-73. PMID: 25535702.
      Citations: 6     Fields:    Translation:Cells
    33. Neudorfer C, Seddik A, Shanab K, Jurik A, Rami-Mark C, Holzer W, Ecker G, Mitterhauser M, Wadsak W, Spreitzer H. Synthesis and in silico evaluation of novel compounds for PET-based investigations of the norepinephrine transporter. Molecules. 2015 Jan 20; 20(1):1712-30. PMID: 25608857.
      Citations:    Fields:    Translation:Humans
    34. Neudorfer C, Shanab K, Jurik A, Schreiber V, Neudorfer C, Vraka C, Schirmer E, Holzer W, Ecker G, Mitterhauser M, Wadsak W, Spreitzer H. Development of potential selective and reversible pyrazoline based MAO-B inhibitors as MAO-B PET tracer precursors and reference substances for the early detection of Alzheimer's disease. Bioorg Med Chem Lett. 2014 Sep 15; 24(18):4490-4495. PMID: 25127869.
      Citations: 2     Fields:    Translation:HumansCells
    35. Palka B, Di Capua A, Anzini M, Vilkauskaité G, Sackus A, Holzer W. Synthesis of trifluoromethyl-substituted pyrazolo[4,3-c]pyridines - sequential versus multicomponent reaction approach. Beilstein J Org Chem. 2014; 10:1759-64. PMID: 25161734.
      Citations: 2     
    36. Shanab K, Neudorfer C, Holzer W, Mitterhauser M, Wadsak W, Spreitzer H. A one-step microwave-assisted synthetic method for an O/S-chemoselective route to derivatives of the first adenosine A3 PET radiotracer. Molecules. 2014 Apr 02; 19(4):4076-82. PMID: 24699149.
      Citations:    Fields:    Translation:Humans
    37. Tarabová D, Soralová S, Breza M, Fronc M, Holzer W, Milata V. Use of activated enol ethers in the synthesis of pyrazoles: reactions with hydrazine and a study of pyrazole tautomerism. Beilstein J Org Chem. 2014; 10:752-60. PMID: 24778729.
      Citations: 3     
    38. Alcántara AR, Pace V, Hoyos P, Sandoval M, Holzer W, Hernáiz MJ. Chemoenzymatic synthesis of carbohydrates as antidiabetic and anticancer drugs. Curr Top Med Chem. 2014; 14(23):2694-711. PMID: 25515749.
      Citations:    Fields:    Translation:HumansAnimalsCells
    39. Pace V, Castoldi L, Holzer W. Addition of lithium carbenoids to isocyanates: a direct access to synthetically useful N-substituted 2-haloacetamides. Chem Commun (Camb). 2013 Sep 28; 49(75):8383-5. PMID: 23938607.
      Citations: 7     Fields:    
    40. Mulla D, Kracher D, Ludwig R, Nagy G, Grandits M, Holzer W, Saber Y, Gabra N, Viernstein H, Unger FM. Azido derivatives of cellobiose: oxidation at C1 with cellobiose dehydrogenase from Sclerotium rolfsii. Carbohydr Res. 2013 Dec 15; 382:86-94. PMID: 24211370.
      Citations:    Fields:    Translation:AnimalsCells
    41. Leepasert T, Shahabi M, Shanab K, Schirmer E, Holzer W, Spreitzer H, Aicher B, Müller G, Günther E. Synthesis and antiproliferative activity of new cytotoxic tri- and tetraazabenzo[3,2-a]fluorene-5,6-dione derivatives. Bioorg Med Chem Lett. 2013 Oct 01; 23(19):5264-6. PMID: 23988351.
      Citations:    Fields:    Translation:HumansCells
    42. Pace V, Castoldi L, Holzer W. Synthesis of a,ß-unsaturated a'-haloketones through the chemoselective addition of halomethyllithiums to Weinreb amides. J Org Chem. 2013 Aug 02; 78(15):7764-70. PMID: 23805887.
      Citations: 6     Fields:    Translation:Cells
    43. Pace V, Hoyos P, Alcántara AR, Holzer W. Chemoselective CaO-mediated acylation of alcohols and amines in 2-methyltetrahydrofuran. ChemSusChem. 2013 May; 6(5):905-10. PMID: 23532956.
      Citations: 1     Fields:    Translation:Cells
    44. Pace V, Vilkauskaite G, Šackus A, Holzer W. Highly efficient and chemoselective a-iodination of acrylate esters through Morita-Baylis-Hillman-type chemistry. Org Biomol Chem. 2013 Feb 21; 11(7):1085-8. PMID: 23303274.
      Citations: 1     Fields:    Translation:Cells
    45. Shahabi M, Schirmer E, Shanab K, Leepasert T, Ruzicka J, Holzer W, Spreitzer H, Aicher B, Schmidt P, Blumenstein L, Müller G, Günther E. Synthesis and biological evaluation of new cytotoxic indazolo[4,3-gh]isoquinolinone derivatives. Bioorg Med Chem Lett. 2013 Mar 15; 23(6):1846-52. PMID: 23395656.
      Citations:    Fields:    Translation:HumansCells
    46. Holzer W, Vilkauskaite G, Arbaciauskiene E, Sackus A. Dipyrazolo[1,5-a:4',3'-c]pyridines - a new heterocyclic system accessed via multicomponent reaction. Beilstein J Org Chem. 2012; 8:2223-9. PMID: 23365633.
      Citations: 2     
    47. Shanab K, Schirmer E, Wulz E, Weissenbacher B, Lassnig S, Slanz R, Fösleitner G, Holzer W, Spreitzer H, Schmidt P, Aicher B, Müller G, Günther E. Synthesis and antiproliferative activity of new cytotoxic azanaphthoquinone pyrrolo-annelated derivatives: Part II. Bioorg Med Chem Lett. 2011 May 15; 21(10):3117-21. PMID: 21458262.
      Citations:    Fields:    Translation:HumansCells
    48. Datterl B, Tröstner N, Kucharski D, Holzer W. Heterocyclic analogues of xanthone and xanthione. 1H-pyrano[2,3-c:6,5-c]dipyrazol-4(7H)-ones and thiones: synthesis and NMR data. Molecules. 2010 Sep 01; 15(9):6106-26. PMID: 20877210.
      Citations: 1     Fields:    
    49. Singh P, Kaur M, Holzer W. Synthesis and evaluation of indole, pyrazole, chromone and pyrimidine based conjugates for tumor growth inhibitory activities--development of highly efficacious cytotoxic agents. Eur J Med Chem. 2010 Nov; 45(11):4968-82. PMID: 20810192.
      Citations: 5     Fields:    Translation:HumansCells
    50. Huemer V, Eller GA, Holzer W. Heterocyclic analogs of xanthiones: 5,6-fused 3-methyl-1-phenylpyrano[2,3-c]pyrazol-4(1H) thiones-synthesis and NMR ((1)H, (13)C, (15)N) data. Magn Reson Chem. 2010 Jun; 48(6):476-82. PMID: 20474027.
      Citations: 1     Fields:    
    51. Shanab K, Schirmer E, Knafl H, Wulz E, Holzer W, Spreitzer H, Schmidt P, Aicher B, Müller G, Günther E. Synthesis and biological evaluation of new cytotoxic azanaphthoquinone pyrrolo-annelated derivatives. Bioorg Med Chem Lett. 2010 Jul 01; 20(13):3950-2. PMID: 20537894.
      Citations:    Fields:    Translation:HumansCells
    52. Fuchs FC, Eller GA, Holzer W. Heterocyclic analogs of thioflavones: synthesis and NMR spectroscopic investigations. Molecules. 2009 Sep 25; 14(9):3814-32. PMID: 19783958.
      Citations: 1     Fields:    
    53. Holzer W, Eller GA, Datterl B, Habicht D. Derivatives of pyrazinecarboxylic acid: 1H, 13C and 15N NMR spectroscopic investigations. Magn Reson Chem. 2009 Jul; 47(7):617-24. PMID: 19402051.
      Citations: 2     Fields:    
    54. Holzer W, Claramunt RM, López C, Alkorta I, Elguero J. A study in desmotropy. Solid State Nucl Magn Reson. 2008 Jul-Sep; 34(1-2):68-76. PMID: 18804750.
      Citations: 1     Fields:    
    55. Singh P, Mittal A, Kaur S, Holzer W, Kumar S. 2, 3-Diaryl-5-ethylsulfanylmethyltetrahydrofurans as a new class of COX-2 inhibitors and cytotoxic agents. Org Biomol Chem. 2008 Aug 07; 6(15):2706-12. PMID: 18633528.
      Citations: 1     Fields:    Translation:HumansCells
    56. Shanab K, Pongprom N, Wulz E, Holzer W, Spreitzer H, Schmidt P, Aicher B, Müller G, Günther E. Synthesis and biological evaluation of novel cytotoxic azanaphthoquinone annelated pyrrolo oximes. Bioorg Med Chem Lett. 2007 Nov 15; 17(22):6091-5. PMID: 17904839.
      Citations: 3     Fields:    Translation:HumansCells
    57. Eller G, Holzer W. A convenient approach to heterocyclic building blocks: synthesis of novel ring systems containing a [5,6]Pyrano[2,3-c]pyrazol-4(1H)-one moiety. Molecules. 2007 Jan 26; 12(1):60-73. PMID: 17693953.
      Citations: 2     Fields:    Translation:Cells
    58. Eller GA, Holzer W. First synthesis of 3-acetyl-2-aminothiophenes using the Gewald reaction. Molecules. 2006 May 16; 11(5):371-6. PMID: 17962769.
      Citations: 4     Fields:    
    59. Singh P, Paul K, Holzer W. Synthesis of pyrazole-based hybrid molecules: search for potent multidrug resistance modulators. Bioorg Med Chem. 2006 Jul 15; 14(14):5061-71. PMID: 16554161.
      Citations: 2     Fields:    Translation:Humans
    60. Singh P, Paul K, Holzer W. Synthesis of 5-acyl-6-[2-hydroxy-3-(amino)propylamino]-1,3-dialkyl-1H-pyrimidine-2,4-diones. Org Biomol Chem. 2005 Nov 07; 3(21):3958-65. PMID: 16240014.
      Citations:    Fields:    Translation:Cells
    61. Holzer W, Claramunt RM, Pérez-Torralba M, Guggi D, Brehmer TH. Spiro-fused (C2)-azirino-(C4)-pyrazolones, a new heterocyclic system. Synthesis, spectroscopic studies and X-ray structure analysis. J Org Chem. 2003 Oct 17; 68(21):7943-50. PMID: 14535769.
      Citations: 1     Fields:    
    62. Ecker GF, Csaszar E, Kopp S, Plagens B, Holzer W, Ernst W, Chiba P. Identification of ligand-binding regions of P-glycoprotein by activated-pharmacophore photoaffinity labeling and matrix-assisted laser desorption/ionization-time-of-flight mass spectrometry. Mol Pharmacol. 2002 Mar; 61(3):637-48. PMID: 11854445.
      Citations: 9     Fields:    Translation:HumansCells