"Thiadiazoles" is a descriptor in the National Library of Medicine's controlled vocabulary thesaurus,
MeSH (Medical Subject Headings). Descriptors are arranged in a hierarchical structure,
which enables searching at various levels of specificity.
No definition found.
| Descriptor ID |
D013830
|
| MeSH Number(s) |
D02.886.675.867 D03.383.129.708.867
|
| Concept/Terms |
|
Below are MeSH descriptors whose meaning is more general than "Thiadiazoles".
Below are MeSH descriptors whose meaning is more specific than "Thiadiazoles".
This graph shows the total number of publications written about "Thiadiazoles" by people in this website by year, and whether "Thiadiazoles" was a major or minor topic of these publications.
To see the data from this visualization as text,
click here.
| Year | Major Topic | Minor Topic | Total |
|---|
| 1994 | 2 | 0 | 2 |
| 1995 | 2 | 0 | 2 |
| 1997 | 1 | 0 | 1 |
| 1999 | 2 | 0 | 2 |
| 2000 | 1 | 0 | 1 |
| 2001 | 0 | 1 | 1 |
| 2002 | 10 | 0 | 10 |
| 2003 | 7 | 1 | 8 |
| 2004 | 4 | 5 | 9 |
| 2005 | 16 | 7 | 23 |
| 2006 | 15 | 9 | 24 |
| 2007 | 25 | 6 | 31 |
| 2008 | 18 | 6 | 24 |
| 2009 | 22 | 9 | 31 |
| 2010 | 33 | 13 | 46 |
| 2011 | 34 | 13 | 47 |
| 2012 | 43 | 12 | 55 |
| 2013 | 28 | 20 | 48 |
| 2014 | 36 | 12 | 48 |
| 2015 | 35 | 12 | 47 |
| 2016 | 43 | 18 | 61 |
| 2017 | 37 | 29 | 66 |
| 2018 | 27 | 17 | 44 |
| 2019 | 18 | 4 | 22 |
| 2020 | 2 | 0 | 2 |
To return to the timeline, click here.
Below are the most recent publications written about "Thiadiazoles" by people in Profiles.
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Highly Potent and Selective Ectonucleoside Triphosphate Diphosphohydrolase (ENTPDase1, 2, 3 and 8) Inhibitors Having 2-substituted-7- trifluoromethyl-thiadiazolopyrimidones Scaffold. Med Chem. 2020; 16(5):689-702.
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Design, Synthesis, Molecular Docking Study and Anti-Hepatocellular Carcinoma Evaluation of New Bis-Triazolothiadiazines. Mini Rev Med Chem. 2020; 20(9):788-800.
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Treatment of Menopausal Vasomotor Symptoms With Fezolinetant, a Neurokinin 3 Receptor Antagonist: A Phase 2a Trial. J Clin Endocrinol Metab. 2019 12 01; 104(12):5893-5905.
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Design, synthesis, and anticancer evaluation of novel quinoline derivatives of ursolic acid with hydrazide, oxadiazole, and thiadiazole moieties as potent MEK inhibitors. J Enzyme Inhib Med Chem. 2019 Dec; 34(1):955-972.
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Design, synthesis, in vitro evaluation, molecular docking and ADME properties studies of hybrid bis-coumarin with thiadiazole as a new inhibitor of Urease. Bioorg Chem. 2019 11; 92:103235.
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Low molecular weight PEG-PLGA polymers provide a superior matrix for conjugated polymer nanoparticles in terms of physicochemical properties, biocompatibility and optical/photoacoustic performance. J Mater Chem B. 2019 09 07; 7(33):5115-5124.
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Effect of benzothiadiazole treatment on improving the mitochondrial energy metabolism involved in induced resistance of apple fruit during postharvest storage. Food Chem. 2020 Jan 01; 302:125288.
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Discovery of a Thiadiazole-Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models. J Med Chem. 2019 07 25; 62(14):6540-6560.
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2,5-Disubstituted thiadiazoles as potent ß-glucuronidase inhibitors; Synthesis, in vitro and in silico studies. Bioorg Chem. 2019 10; 91:103126.
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2-(Bipiperidin-1-yl)-5-(nitroaryl)-1,3,4-thiadiazoles: Synthesis, evaluation of in vitro leishmanicidal activity, and mechanism of action. Bioorg Med Chem. 2019 08 15; 27(16):3682-3691.